Daraxonrasib API / RMC-6236
Research context: RAS(ON) multi-selective inhibitor.
Open primary source↗
APIs & formulation materialsSource-first knowledge base
Primary regulatory records, compound data, clinical trials and peer-reviewed sources for Daraxonrasib, Vopimetostat, Zoldonrasib and Silevertinib.
Editorial standard
Medical and regulatory information changes. We prioritize FDA, NCBI, ClinicalTrials.gov and original peer-reviewed publications, show review dates on medical explainers and separate Daraxon product statements from independently published evidence.
Research context: RAS(ON) multi-selective inhibitor.
Open primary source↗Research context: PRMT5 / MTAP-deleted cancers.
Open primary source↗Research context: RAS(ON) G12D-selective inhibitor.
Open primary source↗Research context: EGFR-mutant NSCLC / EGFR-altered glioblastoma.
Open primary source↗Official approval notice identifying RASONQUE, its active ingredient, sponsor and approved population.
Open primary source↗FDA’s annual list records Rasonque (daraxonrasib) and the approval date.
Open primary source↗FDA 2026 Q3 records: Daraxonrasib 43871, Vopimetostat 44318, Zoldonrasib 44304 and Silevertinib 44854. All four are Type II, status A, under SHANGHAI DA'AN XIN BIOMEDICAL CO LTD.
Open primary source↗Chemical formula, molecular weight, CAS identifier, structure and synonyms.
Open primary source↗Foundational work describing the active-state RAS tri-complex strategy.
Open primary source↗Preclinical characterization and initial clinical translation of RMC-6236.
Open primary source↗Phase 1–2 clinical report focused on previously treated RAS-mutated PDAC.
Open primary source↗Peer-reviewed phase 3 RASolute 302 report.
Open primary source↗Study record for RMC-6236 in advanced solid tumors with specified RAS mutations.
Open primary source↗Phase 3 record in previously treated metastatic pancreatic ductal adenocarcinoma.
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